PAR2 Inhibitor
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FSLLRY-NH2
0 ImagesFSLLRY-NH2 is a protease-activated receptor 2 (PAR2) inhibitor.
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KLK5-IN-1
0 ImagesCat. No.: HY-P11840KLK5-IN-1 is a selective kallikrein 5 (KLK5) inhibitor with an IC50 of 14 nM and a Ki of 11 nM. KLK5-IN-1 reduces KLK5-mediated PAR2-dependent calcium mobilization. KLK5-IN-1 improves epithelial barrier integrity. KLK5-IN-1 can be used in research related to atopic dermatitis and Netherton syndrome.
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I-287
0 ImagesI-287 is a orally active selective PAR2 inhibitor that acting as a negative allosteric regulator on Gαq and Gα12/13 activity and their downstream effectors. I-287 reduces Complete Freund's adjuvant (HY-153808)-induced inflammation in mice and can be used for inflammation/immunology research.
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FSLLRY-NH2 TFA
0 ImagesCat. No.: HY-P1260APurity: 98.97%FSLLRY-NH2 TFA is a protease-activated receptor 2 (PAR2) inhibitor.
